The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Feb. 03, 2015

Filed:

Dec. 06, 2012
Applicant:

Wisconsin Alumni Research Foundation, Madison, WI (US);

Inventors:

Arnold E. Ruoho, Madison, WI (US);

Abdol R. Hajipour, Madison, WI (US);

Uyen B. Chu, Madison, WI (US);

Dominique A. Fontanilla, Twickenham, GB;

Assignee:
Attorneys:
Primary Examiner:
Int. Cl.
CPC ...
A01N 33/02 (2006.01); A61K 31/135 (2006.01); A01N 33/26 (2006.01); A61K 31/655 (2006.01); C07C 247/00 (2006.01); C07J 41/00 (2006.01); C07C 211/00 (2006.01); C12N 5/00 (2006.01); C12N 5/02 (2006.01); C07C 247/16 (2006.01); C07C 211/27 (2006.01); C07C 211/29 (2006.01); C07C 211/49 (2006.01);
U.S. Cl.
CPC ...
C07C 247/16 (2013.01); C07C 211/27 (2013.01); C07C 211/29 (2013.01); C07C 211/49 (2013.01);
Abstract

The invention provides compounds of the formulas described herein and compositions thereof. The invention further provides methods of using the compounds and compositions. The compounds of the invention can provide high affinity binding to sigma-1 receptors in a mammal. The compounds can exhibit selectivity for the sigma-1 receptor over the sigma-2 receptor. The compounds and compositions of the invention can also be used to treat conditions that involve the sigma-1 receptor, such as addiction, cardiovascular conditions, and cancer, for example, cancer of the breast, lung, prostate, ovarian, colorectal, or the CNS.


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