The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Dec. 30, 2014

Filed:

Jun. 07, 2011
Applicants:

David Fairlie, Mt. Ommaney, AU;

Rosemary Sharon Harrison, Bondi Junction, AU;

Nicholas Evan Shepherd, Blackburn North, AU;

Inventors:

David Fairlie, Mt. Ommaney, AU;

Rosemary Sharon Harrison, Bondi Junction, AU;

Nicholas Evan Shepherd, Blackburn North, AU;

Assignee:
Attorney:
Primary Examiner:
Assistant Examiner:
Int. Cl.
CPC ...
A61K 38/10 (2006.01); A61K 45/06 (2006.01); C07K 7/08 (2006.01); A61P 11/00 (2006.01); A61P 11/06 (2006.01); A61P 11/16 (2006.01); A61P 13/00 (2006.01); A61P 13/02 (2006.01); A61P 15/00 (2006.01); A61P 15/10 (2006.01); A61P 1/00 (2006.01); A61P 25/00 (2006.01); A61K 38/12 (2006.01); C07K 7/60 (2006.01); A61K 38/00 (2006.01);
U.S. Cl.
CPC ...
A61K 38/10 (2013.01); A61K 38/00 (2013.01); A61K 45/06 (2013.01); A61K 38/12 (2013.01); C07K 7/08 (2013.01); C07K 7/60 (2013.01);
Abstract

The present invention relates to nociceptin peptide mimetics that have α-helical structures and bind to and modulate the opioid receptor-like-1 (ORL-1) receptor. The peptide mimetics are constrained cyclic nociceptin analogs which have either agonist or antagonist activity. Pharmaceutical compositions comprising the nociceptin peptide mimetics and methods of treating or preventing a disease or condition ameliorated by modulating the ORL-1 receptor are also described.


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