The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Dec. 02, 2014

Filed:

Mar. 15, 2012
Applicants:

Steven Staben, South San Francisco, CA (US);

Jianwen Feng, South San Francisco, CA (US);

Pui Leng Loke, Abingdon, GB;

Christian A. G. N. Montalbetti, Abingdon, GB;

Inventors:

Steven Staben, South San Francisco, CA (US);

Jianwen Feng, South San Francisco, CA (US);

Pui Leng Loke, Abingdon, GB;

Christian A. G. N. Montalbetti, Abingdon, GB;

Assignee:

Genentech, Inc., South San Francisco, CA (US);

Attorneys:
Int. Cl.
CPC ...
C07D 401/14 (2006.01); C07D 403/04 (2006.01); C07D 405/14 (2006.01); C07D 413/14 (2006.01); C07D 417/14 (2006.01); C07D 487/04 (2006.01); A61K 31/506 (2006.01); A61K 31/53 (2006.01); A61K 31/4184 (2006.01); A61P 19/02 (2006.01); C07D 403/14 (2006.01); C07D 491/10 (2006.01);
U.S. Cl.
CPC ...
C07D 417/14 (2013.01); C07D 401/14 (2013.01); C07D 403/04 (2013.01); C07D 403/14 (2013.01); C07D 405/14 (2013.01); C07D 413/14 (2013.01); C07D 487/04 (2013.01); C07D 491/10 (2013.01);
Abstract

The invention relates to novel compounds of Formula I: wherein A, Y, R, Rand the subscript b each has the meaning as described herein and compounds of Formula I, and stereoisomers, geometric isomers, tautomers, solvates, metabolites, isotopes, pharmaceutically acceptable salts, or prodrugs thereof. Compounds of Formula I and pharmaceutical compositions thereof are useful in the treatment of disease and disorders in which undesired or over-activation of NF-kB signaling is observed.


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