The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.
The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.
Patent No.:
Date of Patent:
Oct. 14, 2014
Filed:
Apr. 29, 2011
Applicant:
David J. Fairfax, Slingerlands, NY (US);
Inventor:
David J. Fairfax, Slingerlands, NY (US);
Assignee:
Kinentia Biosciences LLC, Rensselaer, NY (US);
Primary Examiner:
Int. Cl.
CPC ...
C07D 211/08 (2006.01); A61K 31/485 (2006.01); C07D 489/02 (2006.01); C07D 491/18 (2006.01); C07D 405/06 (2006.01); C07D 211/38 (2006.01); A61K 31/445 (2006.01); C07D 489/08 (2006.01); C07D 221/06 (2006.01); C07D 471/08 (2006.01);
U.S. Cl.
CPC ...
A61K 31/445 (2013.01); A61K 31/485 (2013.01); C07D 489/02 (2013.01); C07D 491/18 (2013.01); C07D 405/06 (2013.01); C07D 211/38 (2013.01); C07D 489/08 (2013.01); C07D 221/06 (2013.01); C07D 471/08 (2013.01);
Abstract
4-Fluoro-4-phenylpiperidin-1-yl μ antagonists of general structure as well as pharmaceutical compositions comprising compounds of formula I, are disclosed. These compounds and compositions are useful as treatments of conditions or diseases associated with binding opioid receptors including pain, obesity, hyperalgesia, inflammation, osteoarthritis, drug addiction, and cancer. These compounds and compositions are also useful as treatments for tardive dyskinesia.