The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Oct. 14, 2014

Filed:

Apr. 26, 2011
Applicants:

Floris Louis Van Delft, Nijmegen, NL;

Floris Petrus Johannes Theodorus Rutjes, Wijchen, NL;

Frederik Jan Dommerholt, Beuningen, NL;

Inventors:
Assignee:

Synaffix B.V., Oss, NL;

Attorneys:
Primary Examiner:
Assistant Examiner:
Int. Cl.
CPC ...
C07C 33/16 (2006.01); C07C 271/10 (2006.01); A61K 47/48 (2006.01); A61K 49/00 (2006.01); G01N 33/531 (2006.01); G01N 33/68 (2006.01); G01N 33/58 (2006.01); C07C 271/12 (2006.01); G01N 33/532 (2006.01); C07C 67/347 (2006.01); C07C 29/147 (2006.01); C07C 29/62 (2006.01); C07C 29/58 (2006.01);
U.S. Cl.
CPC ...
C07C 33/16 (2013.01); G01N 33/585 (2013.01); C07C 271/12 (2013.01); G01N 33/532 (2013.01); A61K 47/48023 (2013.01); C07C 67/347 (2013.01); A61K 49/0052 (2013.01); C07C 29/147 (2013.01); C07C 29/62 (2013.01); C07C 2102/24 (2013.01); C07C 29/58 (2013.01);
Abstract

The invention relates to fused cyclooctyne compounds, and to a method for their preparation. The invention also relates to a conjugate wherein a fused cyclooctyne compound according to the invention is conjugated to a label, and to the use of these conjugates in bioorthogonal labeling, imaging and/or modification, such as for example surface modification, of a target molecule. The invention further relates to a method for the modification of a target molecule, wherein a conjugate according to the invention is reacted with a compound comprising a 1,3-dipole or a 1,3-(hetero)diene.


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