The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.
The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.
Patent No.:
Date of Patent:
Oct. 07, 2014
Filed:
Apr. 20, 2012
Applicants:
Uwe Heinelt, Wiesbaden, DE;
Volkmar Wehner, Sandberg, DE;
Matthias Herrmann, Hofheim, DE;
Karl Schoenafinger, Alzenau, DE;
Henning Steinhagen, Sulzbach, DE;
Inventors:
Uwe Heinelt, Wiesbaden, DE;
Volkmar Wehner, Sandberg, DE;
Matthias Herrmann, Hofheim, DE;
Karl Schoenafinger, Alzenau, DE;
Henning Steinhagen, Sulzbach, DE;
Assignee:
Sanofi, Paris, FR;
Attorney:
Primary Examiner:
Assistant Examiner:
Int. Cl.
CPC ...
C07D 249/00 (2006.01); C07D 413/06 (2006.01); C07D 487/04 (2006.01); C07D 471/04 (2006.01); A61P 7/00 (2006.01);
U.S. Cl.
CPC ...
C07D 487/04 (2013.01); C07D 471/04 (2013.01);
Abstract
The invention relates to novel compounds of formula I where X, A, Q1, Q2, Q3, R2, R3, R4, R5, R6, R7, R8 and R9 are each as defined below. The compounds of formula I have antithrombotic activity and inhibit especially protease-activated receptor 1 (PAR1). The invention further relates to a process for preparing the compound of formula I and to the use thereof as a medicament.