The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Sep. 30, 2014

Filed:

Mar. 13, 2013
Applicant:

University of Southern California, Los Angeles, CA (US);

Inventors:

Lin Chen, La Canada, CA (US);

Nimanthi Jayathilaka, Los Angeles, CA (US);

Aidong Han, Los Angeles, CA (US);

Nicos A. Petasis, Hacienda Heights, CA (US);

Assignee:

University of Southern California, Los Angeles, CA (US);

Attorney:
Primary Examiner:
Assistant Examiner:
Int. Cl.
CPC ...
C07D 213/00 (2006.01); C07D 213/40 (2006.01); C07C 233/43 (2006.01); A61K 31/444 (2006.01); A61K 31/00 (2006.01); G01N 33/68 (2006.01); A61K 31/167 (2006.01);
U.S. Cl.
CPC ...
C07C 233/43 (2013.01); C07D 213/40 (2013.01); A61K 31/444 (2013.01); C07K 2299/00 (2013.01); A61K 31/00 (2013.01); G01N 33/6875 (2013.01); G01N 2500/00 (2013.01); A61K 31/167 (2013.01);
Abstract

Disclosed are methods and compositions for modulating the function of transcription factors, especially transcription factors that recruit epigenetic regulators (histone modifying enzymes) to specific DNA promoters. The targeted transcription factors include but are not limited to the myocyte enhancing factor (MEF2), the forkhead/winged helix transcription factor FOXP3 and the transcription factor GATA3. Also disclosed are small molecule modulators of MEF2 and its associated factors that include but not limited to histone deacetylases (HDACs), p300/CBP and Cabin1 and the therapeutic applications thereof.


Find Patent Forward Citations

Loading…