The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.
The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.
Patent No.:
Date of Patent:
Sep. 09, 2014
Filed:
Dec. 13, 2011
Alexandre Vasilievich Ivachtchenko, Encinitas, CA (US);
Oleg Dmitrievich Mitkin, Khimki, RU;
Madina Georgievna Kadieva, Podosinki, RU;
Alexandre Vasilievich Ivachtchenko, Encinitas, CA (US);
Oleg Dmitrievich Mitkin, Khimki, RU;
Madina Georgievna Kadieva, Podosinki, RU;
Other;
Abstract
The present invention relates to novel substituted methyl-amines, serotonin 5-HTreceptor antagonists, to active components, pharmaceutical compositions, method for prophylaxis and treatment of CNS diseases and 'molecular tools', in which novel substituted methyl-amines represent compounds of the general formula 1 and their crystalline forms and pharmaceutically acceptable salts, wherein: W represents benzene, naphthalene, indolizine, quinoline or oxazole cycle; R1=H, F, Cl; R2 represents hydrogen, fluoro, methyl, phenyl, thienyl, furan-2-yl, pyridyl, piperazin-1-yl or 4-methylpiperazin-1-yl; R3 represents cyclopropyl or optionally substituted methyl; with the exception of the compounds in which W simultaneously represents oxazole cycle and R2=phenyl or pyridyl.