The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Patent No.:

US 8791294 B1

PDF
Full Text
Expired
Date of Patent:
Jul. 29, 2014

Filed:

Nov. 19, 2008
Applicants:

Llorenç Rafecas Jane, Tarragona, ES;

Antoni Riera Escale, Barcelona, ES;

Rosario Ramon Albalate, Barcelona, ES;

Monica Alonso Xalma, Barcelona, ES;

Inventors:

Llorenç Rafecas Jane, Tarragona, ES;

Antoni Riera Escale, Barcelona, ES;

Rosario Ramon Albalate, Barcelona, ES;

Monica Alonso Xalma, Barcelona, ES;

Assignee:

BCN Peptides, S.A., Barcelona, ES;

Attorney:
Primary Examiner:
Int. Cl.
CPC ...
C07C 229/36 (2006.01); C07K 5/087 (2006.01);
U.S. Cl.
CPC ...
Abstract

The invention relates to a process for the stereoselective preparation of amino acid derivatives, comprising a hydrogenation reaction of the compound of formula (III), alternatively its enantiomer, wherein R is (C-C)-alkyl; followed by a hydrolysis reaction to obtain L-mesityl alanine, alternatively its enantiomer D-mesityl alanine and, optionally, subjecting said compound to an amino group protection reaction, particularly as Fmoc. It also comprises Fmoc-L- or Fmoc-D-mesityl alanine as products per se, useful as intermediates in preparing peptides or peptide analogs with therapeutic or biological activity.


Find Patent Forward Citations

Rafecas Jane, Llorenç. (2014). Method for the stereoselective preparation of amino acid derivatives (U.S. Patent No. 8791294). U.S. Patent and Trademark Office. https://idiyas.com/patent/badge/8791294

Data source: USPTO (United States Patent and Trademark Office) public patent records. Weekly synchronization. How IDiyas builds this profile

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