The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Jul. 29, 2014

Filed:

Jun. 10, 2009
Applicants:

Ari Melnick, New York, NY (US);

Leandro Cerchietti, New York, NY (US);

Inventors:

Ari Melnick, New York, NY (US);

Leandro Cerchietti, New York, NY (US);

Attorney:
Primary Examiner:
Int. Cl.
CPC ...
A61K 38/04 (2006.01); A61K 38/08 (2006.01); A61K 38/00 (2006.01); C07K 7/06 (2006.01); C07K 7/00 (2006.01); A61K 47/48 (2006.01);
U.S. Cl.
CPC ...
C07K 7/06 (2013.01); C07K 7/00 (2013.01); C07K 2319/00 (2013.01); C07K 2319/10 (2013.01); A61K 38/04 (2013.01); A61K 38/08 (2013.01); A61K 38/00 (2013.01); A61K 47/48315 (2013.01);
Abstract

The invention is directed to a compound that binds to a BCL6 lateral groove and prevents binding of a corepressor to the lateral groove. The present invention is further directed to methods for blocking corepressor binding to a BCL6 lateral groove, methods for inhibiting BCL6 repression in a mammalian cell, and methods for treating a mammal with cancer, wherein the cancer requires BCL6 repression. The present invention is further directed to polypeptides comprising a portion of the corepressor binding site for BCL6 and related polynucleotides and vectors.


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