The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
May. 27, 2014

Filed:

Sep. 09, 2010
Applicants:

Yoshikazu Uto, Chiba, JP;

Hiroshi Karasawa, Tokyo, JP;

Kiyosumi Takaishi, Tokyo, JP;

Inventors:

Yoshikazu Uto, Chiba, JP;

Hiroshi Karasawa, Tokyo, JP;

Kiyosumi Takaishi, Tokyo, JP;

Assignee:
Attorney:
Primary Examiner:
Int. Cl.
CPC ...
C07D 217/06 (2006.01); A61K 31/47 (2006.01);
U.S. Cl.
CPC ...
C07D 217/06 (2013.01); A61K 31/47 (2013.01);
Abstract

The present invention relates to a compound or a pharmacologically acceptable salt thereof having an excellent DGAT inhibitory effect and feeding suppressant effect. The present invention provides a compound represented by the general formula (I), or pharmacologically acceptable salt thereof: [wherein,Rrepresents a phenylaminocarbonyl group that may be substituted with 1 to 5 group(s) independently selected from Substituent Group A, a benzoxazol-2-yl group that may be substituted with 1 to 3 group(s) independently selected from Substituent Group A, or the like; Rindependently represents a C-Calkyl group; Rrepresents a group represented by the formula —C(═O)—O—Ror the like; Rrepresents a hydrogen atom, a C-Calkyl group that may be substituted with 1 to 3 group(s) independently selected from Substituent Group B, or the like; X represents an oxygen atom, a methylene group, or a group represented by the formula —NH—, or the like; L represents a single bond, a methylene group, or the like; . . . represents a single bond or a double bond; m represents 1 or 2; n represents an integer of 0 to 5; Substituent Group A represents a halogen atom, a C-Calkyl group, a C-Chalogenated alkyl group, a C-Calkoxy group, or the like; and Substituent Group B represents a C-Ccycloalkyl group, a phenyl group, a carboxyl group, or the like].


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