The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
May. 06, 2014

Filed:

Nov. 13, 2009
Applicants:

Ahmed Abouabdellah, Paris, FR;

Nathalie Chereze, Paris, FR;

Aude Fayol, Paris, FR;

Mourad Saady, Paris, FR;

Julien Vache, Paris, FR;

Corinne Veronique, Paris, FR;

Philippe Yaiche, Paris, FR;

Inventors:

Ahmed Abouabdellah, Paris, FR;

Nathalie Chereze, Paris, FR;

Aude Fayol, Paris, FR;

Mourad Saady, Paris, FR;

Julien Vache, Paris, FR;

Corinne Veronique, Paris, FR;

Philippe Yaiche, Paris, FR;

Assignee:

Sanofi, Paris, FR;

Attorney:
Primary Examiner:
Int. Cl.
CPC ...
A61K 31/47 (2006.01); A61K 31/497 (2006.01); A61K 31/498 (2006.01); A61K 31/501 (2006.01); A61K 31/502 (2006.01); A61K 31/506 (2006.01);
U.S. Cl.
CPC ...
Abstract

Compound corresponding to general formula (I): in which Ris a hydrogen or fluorine atom or a hydroxyl, cyano, trifluoromethyl, C-alkyl, C-alkoxy or NRRgroup; n is an integer equal to 1, 2 or 3 and m is an integer equal to 1 or 2; A is a covalent bond or a C-alkylene group; Ris a phenyl, pyridinyl, pyridazinyl, pyrimidinyl, pyrazinyl, triazinyl, naphthyl, quinolinyl, isoquinolinyl, phthalazinyl, quinazolinyl, quinoxalinyl, cinnolinyl or naphthyridinyl group, this group being optionally substituted; Ris a hydrogen or fluorine atom, a C-alkyl group or a tritluoromethyl group; Ris a group selected from furanyl, pyrrolyl, thienyl, isothiazolyl, oxazolyl, isoxazolyl, pyrazolyl, oxadiazolyl, thiadiazolyl, imidazole, triazolyl, tetrazolyl, oxazolone, oxazolidinone, isoxazolone, isoxazolidinone, isothiazolone, isothiazolidinone, imidazolone, imidazolidinone, pyrazolone, pyrazolidinone, oxadiazolone, thiadiazolone and triazolone, this group being optionally substituted; in the form of a base or of an addition salt with an acid. Therapeutic use.


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