The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Jan. 07, 2014

Filed:

Nov. 09, 2012
Applicants:

The Regents of the University of California, Oakland, CA (US);

The University of Connecticut, Farmington, CT (US);

Inventors:

Ohyun Kwon, Los Angeles, CA (US);

Gabriel Fenteany, Storrs, CT (US);

Assignees:
Attorney:
Primary Examiner:
Assistant Examiner:
Int. Cl.
CPC ...
C07D 217/22 (2006.01); C07D 221/02 (2006.01); C07D 217/00 (2006.01); C07D 295/00 (2006.01); C07D 401/00 (2006.01);
U.S. Cl.
CPC ...
Abstract

A method for producing libraries of structurally and stereochemically diverse molecules that can be screened for biological or chemical activity. A library of 91 heterocyclic compounds composed of 16 distinct scaffolds was synthesized through a sequence of phosphine-catalyzed ring-forming reactions, Tebbe reactions, Diels-Alder reactions, and, in some cases, hydrolysis to illustrate the methods. Three compounds inhibiting migration of human breast cancer cells are identified from the library.


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