The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Dec. 24, 2013

Filed:

Mar. 09, 2010
Applicants:

Hanbin Shan, Shanghai, CN;

Peng Zhang, Shanghai, CN;

Zhedong Yuan, Shanghai, CN;

Xudong Jiang, Shanghai, CN;

Yu Huang, Shanghai, CN;

Hubo Wang, Shanghai, CN;

Xufeng Cao, Shanghai, CN;

Xingdong Cheng, Shanghai, CN;

Xiong Yu, Shanghai, CN;

Inventors:

Hanbin Shan, Shanghai, CN;

Peng Zhang, Shanghai, CN;

Zhedong Yuan, Shanghai, CN;

Xudong Jiang, Shanghai, CN;

Yu Huang, Shanghai, CN;

Hubo Wang, Shanghai, CN;

Xufeng Cao, Shanghai, CN;

Xingdong Cheng, Shanghai, CN;

Xiong Yu, Shanghai, CN;

Assignee:

Les Laboratories Servier, Suresnes Cedex, FR;

Attorney:
Primary Examiner:
Int. Cl.
CPC ...
A01N 37/18 (2006.01); A61K 31/16 (2006.01); C07C 233/00 (2006.01); C07C 235/00 (2006.01); C07C 237/00 (2006.01); C07C 239/00 (2006.01);
U.S. Cl.
CPC ...
Abstract

The invention provides a new crystalline form of agomelatine, preparation and use thereof. The X-ray powder diffraction diagram of the agomelatine crystalline form shows main peaks at the diffraction angles 2θ 11.13°, 11.82°, 17.49°, 18.29°, 19.48°, 19.72°, 20.50°, 21.76°, 22.54°, 22.97°, 24.56°, 25.36°, 27.16° and 31.93°. Said new crystalline form is characterized by high purity, stability and good reproducibility, and thus is advantageous for the pharmaceutical formulation. In addition, the stability and solubility of said crystalline form are also superior over the several existing crystalline forms.


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