The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Aug. 06, 2013

Filed:

Nov. 29, 2010
Applicants:

Franz-josef Mais, Düsseldorf, DE;

Joachim Rehse, Leichlingen, DE;

Winfried Joentgen, Köln, DE;

Konrad Siegel, Düsseldorf, DE;

Inventors:

Franz-Josef Mais, Düsseldorf, DE;

Joachim Rehse, Leichlingen, DE;

Winfried Joentgen, Köln, DE;

Konrad Siegel, Düsseldorf, DE;

Assignee:

Bayer Intellectual Property GmbH, Monheim am Rhein, DE;

Attorney:
Int. Cl.
CPC ...
C07D 403/04 (2006.01); A61K 31/506 (2006.01); A61P 19/02 (2006.01);
U.S. Cl.
CPC ...
Abstract

The present invention relates to processes for preparing methyl {4,6-diamino-2-[1-(2-fluorobenzyl)-1H-pyrazolo[3,4-b]pyridin-3-yl]pyrimidin-5-yl}carbamate, i.e. the compound of the formula (I) and to a process for purifying the crude product of the formula (I) for use as pharmaceutically active compound, where, for purification, methyl {4,6-diamino-2-[1-(2-fluorobenzyl)-1H-pyrazolo[3,4-b]pyridin-3-yl]pyrimidin-5-yl}carbamate sulphinyldimethane (1:2) of the formula (II) is isolated as intermediate or is generated as intermediate in this purification process, if appropriate present in a mixture.


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