The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.
The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.
Patent No.:
Date of Patent:
Jul. 09, 2013
Filed:
Apr. 02, 2009
Mogens Peter Cherly Nielsen, Roskilde, DK;
Tommy Liljefors, Frederiksberg, DK;
Jakob Alexander Nilsson, Lund, SE;
Olov a Sterner, Malmö, SE;
Mogens Peter Cherly Nielsen, Roskilde, DK;
Tommy Liljefors, Frederiksberg, DK;
Jakob Alexander Nilsson, Lund, SE;
Olov A Sterner, Malmö, SE;
Innovationspatent Sverige AB, Lund, SE;
Abstract
The present invention relates to novel GABA/BzR ligands of the general formulas (I), (II) and (III) wherein Ris selected from the group consisting of hydrogen, halogen, haloalkyl having 1-2 carbon atoms, alkoxy having 1 to 3 carbon atoms in the alkyl chain, alkyl having 1 to 3 carbon atoms, and nitro, and Ris selected from the group consisting of hydrogen, halogen and alkyl having 1 to 2 carbon atoms, as well as the use of these compounds for treating anxiolytic, anticonvulsant, sedative-hypnotic and myorelaxant conditions as well as anxiogenic, somnolytic and convulsant conditions in mammals including pharmaceutical compositions comprising the same.