The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.
The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.
Patent No.:
Date of Patent:
Oct. 16, 2012
Filed:
Mar. 21, 2011
Pierre-etienne Chabrier DE Lassauniere, Paris, FR;
Jeremiah Harnett, Gif sur Yvette, FR;
Dennis Bigg, Gif sur Yvette, FR;
Anne-marie Liberatore, Auffargis, FR;
Jacques Pommier, Paris, FR;
Jacques Lannoy, Bievres, FR;
Christophe Thurieau, Paris, FR;
Pierre-Etienne Chabrier De Lassauniere, Paris, FR;
Jeremiah Harnett, Gif sur Yvette, FR;
Dennis Bigg, Gif sur Yvette, FR;
Anne-Marie Liberatore, Auffargis, FR;
Jacques Pommier, Paris, FR;
Jacques Lannoy, Bievres, FR;
Christophe Thurieau, Paris, FR;
Ipsen Pharma S.A.S., Boulogne Billancourt, FR;
Abstract
The invention relates to thiazole, oxazole, imidazole, isoxazole and isoxazoline derivatives of general formula (I) wherein Het is thiazole, oxazole, imidazole, isoxazole or isoxazoline, n is an integer from 0 to 6, A is notably selected from various optionally substituted aromatic radicals, B is notably hydrogen, alkyl or phenyl, Rand Rare notably independently hydrogen, alkyl or cycloalkyl and Ω is —NRRor —OR, Rand Rare notably independently hydrogen, alkyl, cycloalkyl or —(CH)—COOR, Ris notably alkyl or haloalkyl and Ris notably hydrogen or alkyl. These compounds have advantageous pharmacological properties which allow their use in therapeutics, notably for treating neurodegenerative disorders or pain.