The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.
The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.
Patent No.:
Date of Patent:
Jun. 21, 2011
Filed:
Jul. 03, 2007
Axel Stoit, Weesp, NL;
Hein K. A. C. Coolen, Weesp, NL;
Martina A. W. Van Der Neut, Weesp, NL;
Cornelis G. Kruse, Weesp, NL;
Axel Stoit, Weesp, NL;
Hein K. A. C. Coolen, Weesp, NL;
Martina A. W. Van Der Neut, Weesp, NL;
Cornelis G. Kruse, Weesp, NL;
Solvay Pharmaceuticals B.V., Weesp, NL;
Abstract
Azaindole derivatives of formula (I): wherein the symbols have the meanings given in the specification, are described. These compounds have a combination of partial nicotinic acetylcholine receptor agonism and dopamine reuptake inhibition. The invention also relates to pharmaceutical compositions containing these compounds, to methods for preparing them, methods for preparing novel intermediates useful for their synthesis, methods for preparing compositions, and uses of such compounds and compositions, for example, their use in administering them to patients to achieve a therapeutic effect in disorders in which nicotinic receptors and/or dopamine transporters are involved, or that can be treated via manipulation of those receptors.