The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Apr. 05, 2011

Filed:

Jul. 02, 2007
Applicants:

Pier Giovanni Baraldi, Ferrara, IT;

Pier Andrea Borea, Ferrara, IT;

Pierangelo Geppetti, Ferrara, IT;

Maria Giovanna Pavani, Ferrara, IT;

Francesca Fruttarolo, Ferrara, IT;

Marcello Trevisani, Ferrara, IT;

Inventors:

Pier Giovanni Baraldi, Ferrara, IT;

Pier Andrea Borea, Ferrara, IT;

Pierangelo Geppetti, Ferrara, IT;

Maria Giovanna Pavani, Ferrara, IT;

Francesca Fruttarolo, Ferrara, IT;

Marcello Trevisani, Ferrara, IT;

Assignee:

Pharmeste S.R.L., Ferrara, IT;

Attorney:
Primary Examiner:
Int. Cl.
CPC ...
C07D 217/00 (2006.01); A61K 31/472 (2006.01);
U.S. Cl.
CPC ...
Abstract

The invention provides compounds of formula (I), wherein Y, R, n and X are as defined in the description, a process for their preparation and pharmaceutical compositions containing them. The compounds of formula (I) inhibit the Transient Receptor Potential Vanilloid 1 (TRPV1), which plays a pivotal role in the development of post-inflammatory analgesia, therefore they can be used as analgesic and anti-inflammatory drugs.


Find Patent Forward Citations

Loading…