The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.
The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.
Patent No.:
Date of Patent:
Jan. 25, 2011
Filed:
Apr. 24, 2003
Wim Meutermans, Toowong, AU;
Michael West, Hemmant, AU;
George Adamson, Hampshire, GB;
Giang Thanh Le, Mt. Gravatt, AU;
Nicholas B. Drinnan, Highgate Hill, AU;
Giovanni Abbenante, Sampsonvale, AU;
Bernd Becker, New Farm, AU;
Matthias Grathwohl, Constance, DE;
Premraj Rajaratnam, Eight Mile Plains, AU;
Gerald Tometzki, Manly West, AU;
Wim Meutermans, Toowong, AU;
Michael West, Hemmant, AU;
George Adamson, Hampshire, GB;
Giang Thanh Le, Mt. Gravatt, AU;
Nicholas B. Drinnan, Highgate Hill, AU;
Giovanni Abbenante, Sampsonvale, AU;
Bernd Becker, New Farm, AU;
Matthias Grathwohl, Constance, DE;
Premraj Rajaratnam, Eight Mile Plains, AU;
Gerald Tometzki, Manly West, AU;
Alchemia Limited, Eight Mile Plains, AU;
Abstract
Methods are described for the preparation of combinatorial libraries of potentially biologically active disaccharide compounds. These compounds are variously functionalized, with a view to varying lipid solubility size, function an other properties, with the particular aim of discovering novel drug or drug-like compounds, or compounds with useful properties. The invention provides intermediates, processes and synthetic strategies for the solution or solid phase synthesis of disaccharides, variously functionalized about the sugar ring, including the addition of aromaticity and charge, and the placement of pharmaceutically useful groups and isosteres.