The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.
The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.
Patent No.:
Date of Patent:
Jan. 04, 2011
Filed:
Mar. 29, 2006
Sylvain Celanire, Feigeres, FR;
Patrice Talaga, Watermael-Boitsfort, BE;
Regorius Leurs, Amsterdam, NL;
Frederic Denonne, Brussels, BE;
Henkdrik Timmerman, Oegstgeest, NL;
Florence Lebon, Lillois, BE;
Sylvain Celanire, Feigeres, FR;
Patrice Talaga, Watermael-Boitsfort, BE;
Regorius Leurs, Amsterdam, NL;
Frederic Denonne, Brussels, BE;
Henkdrik Timmerman, Oegstgeest, NL;
Florence Lebon, Lillois, BE;
UCB Pharma, S.A., Brussels, BE;
Abstract
The present invention relates to compounds comprising an oxazoline or thiazoline moiety, processes for preparing them, pharmaceutical compositions comprising said compounds and their uses as H-receptor ligands, (I), wherein Ais CH C(CH) or N; Ris hydrogen or halogen; Ris (II); Ais O or S; Ris hydrogen, halogen, Calkyl or Calkoxy; Ris hydrogen, halogen, Calkyl, Calkoxy, trifluoromethyl or —O—(CH)n-NReach CHin —O—(CH)n-NR12b being optionally substituted by one or two Calkyl; Ris hydrogen or —O—(CH)—NR, each CHin —O—(CH)—NRRbeing optionally substituted by one or two Calkyl, and at least one of Rand Rshould be a —O—(CH)n-NRRgroup.