The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Jul. 13, 2010

Filed:

Jun. 27, 2008
Applicants:

Richard Sedrani, Basel, CH;

Juergen Klaus Maibaum, Weil-Haltingen, DE;

Werner Breitenstein, Basel, CH;

Holger Sellner, Therwil, CH;

Claus Ehrhardt, Lorrach, DE;

Nils Ostermann, Binzen, DE;

Inventors:

Richard Sedrani, Basel, CH;

Juergen Klaus Maibaum, Weil-Haltingen, DE;

Werner Breitenstein, Basel, CH;

Holger Sellner, Therwil, CH;

Claus Ehrhardt, Lorrach, DE;

Nils Ostermann, Binzen, DE;

Assignee:

Novartis AG, Basel, CH;

Attorney:
Primary Examiner:
Assistant Examiner:
Int. Cl.
CPC ...
A01N 43/54 (2006.01); A01N 43/40 (2006.01); C07D 239/42 (2006.01); C07D 401/04 (2006.01); C07D 239/00 (2006.01); C07D 239/02 (2006.01); C07D 211/08 (2006.01); C07D 401/00 (2006.01); C07D 405/00 (2006.01); C07D 409/00 (2006.01); C07D 411/00 (2006.01); C07D 413/00 (2006.01); C07D 417/00 (2006.01); C07D 419/00 (2006.01); C07D 421/00 (2006.01); C07D 211/68 (2006.01); C07D 211/80 (2006.01); C07D 213/02 (2006.01); A61K 31/445 (2006.01);
U.S. Cl.
CPC ...
Abstract

Compounds of the present invention having the formula (I) exhibit inhibitory activity on the natural enzyme renin. Thus, compounds of formula (I) may be employed for the treatment of hypertension, atherosclerosis, unstable coronary syndrome, congestive heart failure, cardiac hypertrophy, cardiac fibrosis, cardiomyopathy postinfarction, unstable coronary syndrome, diastolic dysfunction, chronic kidney disease, hepatic fibrosis, complications resulting from diabetes, such as nephropathy, vasculopathy and neuropathy, diseases of the coronary vessels, restenosis following angioplasty, raised intra-ocular pressure, glaucoma, abnormal vascular growth, hyperaldosteronism, cognitive impairment, alzheimers, dementia, anxiety states and cognitive disorders.


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