The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.
The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.
Patent No.:
Date of Patent:
Jun. 22, 2010
Filed:
Aug. 05, 2005
Kevin Michael Thewlis, Harlow, GB;
Simon Edward Ward, Harlow, GB;
Kevin Michael Thewlis, Harlow, GB;
Simon Edward Ward, Harlow, GB;
Glaxo Group Limited, Greenford, Middlesex, GB;
Abstract
This case discloses compounds of formula (I) wherein Ris Calkyl, haloCalkyl, Calkenyl, amino, monoCalkylamino or diCalkylamino; Rand R, which may be the same or different, are hydrogen, halogen, Calkyl, haloCalkyl, Calkoxy, haloCalkoxy, cyano or amino; each R, which may be the same or different, is Calkyl, halogen, haloCalkyl, Calkoxy, haloCalkoxy, cyano, nitro or amino; p is 0, 1 or 2; each R, which may be the same or different, is Calkyl, halogen, haloCalkyl, Calkoxy, haloCalkoxy, cyano, nitro or amino; q is 0, 1 or 2; Ris —NRSOR, —NRC(═O)R, —NR(C═O)N(R), —(C═O)R, —CHNRSOR, —CHNRC(═O)R, CHNR(C═O)N(R)or —CH(C═O)R; where Rand each R, which may be the same or different, is hydrogen or Calkyl; Rand Rare Calkyl or haloCalkyl; or Rand R, or Rand R, together with the interconnecting atoms, may form a 5- or 6-membered ring; n is 1 or 2; and Rand R, which may be the same or different, are hydrogen, halogen, Calkyl, haloCalkyl, Calkoxy, haloCalkoxy, cyano or amino. It also discloses methods for preparing the compounds and their use in therapy such as treating schizophrenia.