The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.
The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.
Patent No.:
Date of Patent:
May. 26, 2009
Filed:
May. 11, 2005
Yuichi Suzuki, Tsukuba, JP;
Koichi Ito, Tsukuba, JP;
Atsushi Sasaki, Tsukuba, JP;
Koshi Ueno, Tsukuba, JP;
Miyuki Sakai, Tsukuba, JP;
Hiroki Ishihara, Tsukuba, JP;
Atsuhiko Kubota, Tsukuba, JP;
Yuichi Suzuki, Tsukuba, JP;
Koichi Ito, Tsukuba, JP;
Atsushi Sasaki, Tsukuba, JP;
Koshi Ueno, Tsukuba, JP;
Miyuki Sakai, Tsukuba, JP;
Hiroki Ishihara, Tsukuba, JP;
Atsuhiko Kubota, Tsukuba, JP;
Eisai R & D Management Co., Ltd., Tokyo, JP;
Abstract
The present invention relates to a compound represented by the following formula, a pharmacologically acceptable salt thereof, or a use thereof as a pharmaceutical: wherein Rand Rare substituents adjacent to each other, and together with two carbon atoms to each of which they attach, form a 5- to 7-membered non-aromatic carbocyclic group or the like, which may be substituted by 1 to 4 substituents selected from (1) an oxo group, (2) a hydroxyl group, and the like; Rrepresents a hydrogen atom or the like; and Rrepresents a hydrogen atom or the like. This compound has a superior strength of binding to a 5-HT1A receptor and an antagonism to the receptor, and is useful as an agent for treating or preventing lower urinary tract symptoms, and particularly symptoms regarding urinary storage.