The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.
The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.
Patent No.:
Date of Patent:
Dec. 30, 2008
Filed:
Jul. 09, 2007
Pier Giovanni Baraldi, Ferrara, IT;
Pier Andrea Borea, Ferrara, IT;
Pier Giovanni Baraldi, Ferrara, IT;
Pier Andrea Borea, Ferrara, IT;
King Pharmaceuticals Research and Development, Inc., Cary, NC (US);
Abstract
The compounds of the following formula: wherein R, R, Rand A have the meanings given in the specification, are endowed with selective Aadenosine receptor antagonist activity. These compounds can be used in a pharmaceutical composition to treat disorders caused by excessive activation of the Areceptor, or can be used in a diagnostic application to determine the relative binding of other compounds to the Areceptor. The compounds can be labeled, for example with fluorescent or radiolabels, and the labels used in vivo or in vitro to determine the presence of tumor cells which possess a high concentration of adenosine Areceptors.