The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.
The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.
Patent No.:
Date of Patent:
Oct. 14, 2008
Filed:
Jun. 20, 2005
Lyn Howard Jones, Sandwich, GB;
Charles Eric Mowbray, Sandwich, GB;
David Anthony Price, Sandwich, GB;
Matthew Duncan Selby, Sandwich, GB;
Paul Anthony Stupple, Sandwich, GB;
Lyn Howard Jones, Sandwich, GB;
Charles Eric Mowbray, Sandwich, GB;
David Anthony Price, Sandwich, GB;
Matthew Duncan Selby, Sandwich, GB;
Paul Anthony Stupple, Sandwich, GB;
Pfizer Inc, New York, NY (US);
Abstract
This invention relates to pyrazole derivatives of formula (I) or pharmaceutically acceptable salts, solvates or derivative thereofs, wherein R1 to R4 are defined in the description, and to processes for the preparation thereof, intermediates used in their preparation of, compositions containing them and the uses of such derivatives. The compounds of the present invention bind to the enzyme reverse transcriptase and are modulators, especially inhibitors thereof. As such the compounds of the present invention are useful in the treatment of a variety of disorders including those in which the inhibition of reverse transcriptase is implicated. Disorders of interest include those caused by Human Immunodificiency Virus (HIV) and genetically related retroviruses, such as Acquired Immune Deficiency Syndrome (AIDS).