The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Feb. 05, 2008

Filed:

Sep. 21, 2006
Applicants:

Zoran Rankovic, Newhouse, GB;

Jiaqiang Cai, Newhouse, GB;

Inventors:

Zoran Rankovic, Newhouse, GB;

Jiaqiang Cai, Newhouse, GB;

Assignee:

N.V. Organon, Oss, NL;

Attorney:
Int. Cl.
CPC ...
C07D 239/34 (2006.01); C07D 239/38 (2006.01); C07D 239/42 (2006.01); A61K 31/505 (2006.01); A61P 9/10 (2006.01); A61P 19/02 (2006.01); A61P 19/10 (2006.01); A61P 29/00 (2006.01);
U.S. Cl.
CPC ...
Abstract

Disclosed herein are 4-phenyl-6-substituted-pyrimidine-2-carbonitrile derivatives having Formula I, wherein each of the substituents is given the definition as set forth in the specification and claims; or a pharmaceutically acceptable salt thereof. Also disclosed are pharmaceutical compositions comprising these 4-phenyl-6-substituted-pyrimidine-2-carbonitrile derivatives and use of these 4-phenyl-6-substituted-pyrimidine-2-carbonitrile derivatives for the treatment of cathepsin K and cathepsin S related disorders, e.g. osteoporosis, atherosclerosis, inflammation and immune disorders such as rheumatoid arthritis and chronic pain.


Find Patent Forward Citations

Loading…