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The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Patent No.:

US 7323562 B1

PDFFull Text
Date of Patent:
Jan. 29, 2008

Filed:

Sep. 21, 2005

Method of preparing poly(adp-ribose) polymerases inhibitors

Applicants:

Chunrong MA, San Diego, CA (US);

Naresh Nayyar, San Diego, CA (US);

Nebojsa Slobodan Stanković, La Jolla, CA (US);

Inventors:

Chunrong Ma, San Diego, CA (US);

Naresh Nayyar, San Diego, CA (US);

Nebojsa Slobodan Stanković, La Jolla, CA (US);

Assignees:

Agouron Pharmaceuticals, Inc., San Diego, CA (US);

Cancer Research Technology Ltd., London, GB;

Attorneys:

Bryan C. Zielinski

Galina M. Yakovleva

Primary Examiner:

Bruck Kifle

Int. Cl.
CPC ...
C07D 487/06 (2006.01);
U.S. Cl.
CPC ...
Abstract

This invention relates to a new and convergent route to small molecule inhibitors of poly(ADP-ribose) polymerase, such as 8-fluoro-2-{4-[(methylamino)methyl]phenyl}-1,3,4,5-tetrahydro-6H-azepino[5,4,3-cd]indol-6-one, via a key Sonogashira coupling reaction and a CuI-promoted indole formation.

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Ma, Chunrong. (2008). Method of preparing poly(adp-ribose) polymerases inhibitors (U.S. Patent No. 7323562). U.S. Patent and Trademark Office. https://idiyas.com/patent/badge/7323562

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