The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Nov. 13, 2007

Filed:

Feb. 26, 2002
Applicants:

Nobuhiko Fushimi, Matsumoto, JP;

Hideki Fujikura, Matsumoto, JP;

Toshihiro Nishimura, Hotaka-machi, JP;

Kenji Katsuno, Tatusno-machi, JP;

Masayuki Isaji, Shiojiri, JP;

Inventors:

Nobuhiko Fushimi, Matsumoto, JP;

Hideki Fujikura, Matsumoto, JP;

Toshihiro Nishimura, Hotaka-machi, JP;

Kenji Katsuno, Tatusno-machi, JP;

Masayuki Isaji, Shiojiri, JP;

Assignee:
Attorney:
Primary Examiner:
Assistant Examiner:
Int. Cl.
CPC ...
A01N 43/04 (2006.01); A61K 31/70 (2006.01); C07H 17/00 (2006.01);
U.S. Cl.
CPC ...
Abstract

The present invention provides glucopyranosyloxypyrazole derivatives represented by the general formula: wherein R, Rand Rrepresent a hydrogen atom or a halogen atom; Rrepresents a lower alkyl group or a halo(lower alkyl) group; and Rrepresents a hydrogen atom, a lower alkyl group, a lower alkoxy group, a lower alkylthio group, etc., a pharmaceutically acceptable salt thereof or a prodrug thereof., which exert an excellent inhibitory activity in human SGLT2, and therefore are useful as drugs for the prevention or treatment of a disease associated with hyperglycemia such as diabetes, diabetic complications or obesity, pharmaceutically acceptable salts thereof or prodrugs thereof, production intermediates thereof and pharmaceutical uses thereof.


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