The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Jan. 09, 2007

Filed:

Jan. 09, 2003
Applicants:

Robert W. Desimone, Durham, CT (US);

John M. Peterson, Durham, CT (US);

Cheryl Steenstra, Meriden, CT (US);

Yiping Shen, Branford, CT (US);

Linda M. Gustavson, Guilford, CT (US);

Christopher Mach, Fairfield, CT (US);

Alan Hutchison, Madison, CT (US);

Inventors:

Robert W. DeSimone, Durham, CT (US);

John M. Peterson, Durham, CT (US);

Cheryl Steenstra, Meriden, CT (US);

Yiping Shen, Branford, CT (US);

Linda M. Gustavson, Guilford, CT (US);

Christopher Mach, Fairfield, CT (US);

Alan Hutchison, Madison, CT (US);

Assignee:

Neurogen Corporation, Branford, CT (US);

Attorneys:
Primary Examiner:
Int. Cl.
CPC ...
A61P 15/00 (2006.01); A61K 31/55 (2006.01); A61K 31/495 (2006.01); C07D 243/08 (2006.01); C07D 401/00 (2006.01);
U.S. Cl.
CPC ...
Abstract

Melanin concentrating hormone receptor ligands (especially substituted 2-(4-benzyl-piperazin-1-ylmethyl)-1H-benzoimidazole analogues), capable of modulating MCH receptor activity, are provided. Such ligands may be used to modulate MCH binding to MCH receptors in vivo or in vitro, and are particularly useful in the treatment of a variety of metabolic, feeding and sexual disorders in humans, domesticated companion animals and livestock animals. Pharmaceutical compositions and methods for treating such disorders are provided, as are methods for using such ligands for detecting MCH receptors (e.g., receptor localization studies).


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