The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
May. 23, 2006

Filed:

May. 15, 2003
Applicants:

Brian M. Aquila, Marlborough, MA (US);

Seth C. Hopkins, Clinton, MA (US);

Curtis A. Lockshin, Lexington, MA (US);

Fengjiang Wang, Northborough, MA (US);

Inventors:

Brian M. Aquila, Marlborough, MA (US);

Seth C. Hopkins, Clinton, MA (US);

Curtis A. Lockshin, Lexington, MA (US);

Fengjiang Wang, Northborough, MA (US);

Assignee:

Sepracor Inc., Marlborough, MA (US);

Attorneys:
Primary Examiner:
Int. Cl.
CPC ...
A61K 31/135 (2006.01); A61K 31/34 (2006.01); A61K 31/44 (2006.01); C07D 307/04 (2006.01);
U.S. Cl.
CPC ...
Abstract

One aspect of the present invention relates to amines. A second aspect of the present invention relates to the use of the amines as inhibitors of a mammalian anandamide transporter. The compounds of the present invention will also find use in the treatment of numerous ailments, conditions and diseases which afflict mammals, including but not limited to asthma, neuropathic pain, persistent pain, inflammatory pain, hyperactivity, hypertension, brain ischemia, Parkinson's disease, spasticity, Tourette's syndrome, schizophrenia, hemorrhagic shock, septic shock, cardiac shock, migrane, Horton's headache, multiple sclerosis, anorexia, AIDS wasting syndrome, organ rejection, autoimmune diseases, allergy, arthritis, Crohn's disease, malignant gliomas, neurodegenerative diseases, Huntington's chorea, glaucoma, nausea, anxiety, psychosis, attention deficit hyperactivity disorder, premature ejaculation, and stroke. Another aspect of the present invention relates to combinatorial libraries of amines, and methods for preparing the libraries.


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