The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.
The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.
Patent No.:
Date of Patent:
Apr. 25, 2006
Filed:
May. 19, 2004
Takahiko Tobe, Tsukuba, JP;
Takashi Sugane, Tsukuba, JP;
Wataru Hamaguchi, Tsukuba, JP;
Itsuro Shimada, Tsukuba, JP;
Kyoichi Maeno, Tsukuba, JP;
Junji Miyata, Tsukuba, JP;
Tetsuya Kimizuka, Itabashi-ku, JP;
Takeshi Suzuki, Tsukuba, JP;
Atsuyuki Kohara, Tsukuba, JP;
Takuma Morita, Tsukuba, JP;
Michael Arlt, Seeheim Jugenheim, DE;
Hartmut Greiner, Weiterstadt, DE;
Takahiko Tobe, Tsukuba, JP;
Takashi Sugane, Tsukuba, JP;
Wataru Hamaguchi, Tsukuba, JP;
Itsuro Shimada, Tsukuba, JP;
Kyoichi Maeno, Tsukuba, JP;
Junji Miyata, Tsukuba, JP;
Tetsuya Kimizuka, Itabashi-ku, JP;
Takeshi Suzuki, Tsukuba, JP;
Atsuyuki Kohara, Tsukuba, JP;
Takuma Morita, Tsukuba, JP;
Michael Arlt, Seeheim Jugenheim, DE;
Hartmut Greiner, Weiterstadt, DE;
Astellas Pharma, Inc., Tokyo, JP;
Abstract
The invention relates to a triazole derivative with an activity inhibiting glycine transporter and for use as a pharmaceutical drug, and a novel triazole derivative. The inventive triazole derivative has an excellent activity inhibiting glycine transporter and is useful as a therapeutic agent of dementia, schizophrenia, cognitive disorders, or cognitive disorders involved in various diseases such as Alzheimer disease, Parkinson's disease, or Huntington disease or the like, or spasm involved in diseases such as nerve degenerative diseases and cerebrovascular disorders, or the like. Particularly, the pharmaceutical drug is useful for the amelioration of learning disability of dementia and the like.