The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Apr. 25, 2006

Filed:

Dec. 20, 2000
Applicants:

Matthias Gerlach, Brachttal, DE;

Corinna Maul, Aachen, DE;

Inventors:

Matthias Gerlach, Brachttal, DE;

Corinna Maul, Aachen, DE;

Assignee:

Gruenenthal GmbH, Aachen, DE;

Attorney:
Primary Examiner:
Int. Cl.
CPC ...
A61K 31/535 (2006.01); C07D 207/00 (2006.01);
U.S. Cl.
CPC ...
Abstract

The invention relates to substituted pyrrole Mannich bases of general formula (I), wherein R=H, a C-alkyl-, aryl, a heteroaryl- or an aryl, heteroaryl-, CN, Br—, Cl or OH radical bound by a Calkylene group, R=CH(R)N(R)(R), R3, R3', R3″ identically or individually represent H, F, Cl, Br, CF, CN, NO, SONH, NHR, SR, OR, CO(OR), CHCO(OR), COR, a C-alkyl-, aryl-, heteroaryl-aryl radical or a heteroalkyl radical bound by a Calkylene group, R=an unsubstituted phenyl radical or a phenyl radical substituted at least with Calkyl, C-alkoxy-, halogen-, a method for the production of the above-mentioned compounds, medicaments containing said compounds, and the use of said compounds in the production of medicaments. Said active ingredients are particularly suitable for pain therapy, and for treating inflammatory and allergic reactions, drug or alcohol abuse, diarrhoea, gastritis, ulcers, cardiovascular diseases, urinary incontinence, depressions, states of shock, migranes, narcolepsy, overweight, asthma, glaucoma, hyperkinetic syndrome, lack of drive, bulimia, anorexia, catalepsia, anxiolysis increasing vigilance and/or increasing libido.


Find Patent Forward Citations

Loading…