The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.
The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.
Patent No.:
Date of Patent:
Apr. 29, 2003
Filed:
Jul. 20, 2001
Applicant:
Inventors:
Rodney L. Parsons, Wilmington, DE (US);
Roberta L. Dorow, Portage, MI (US);
Akin H. Davulcu, Wilmington, DE (US);
Joseph M. Fortunak, Hawthorn Woods, IL (US);
Gregory D. Harris, Wilmington, DE (US);
Goss S. Kauffman, Bear, DE (US);
William A. Nugent, Wilmington, DE (US);
Lilian A. Radesca, Newark, DE (US);
Assignee:
Bristol-Myers Squibb Pharma, Princeton, NJ (US);
Attorney:
Primary Examiner:
Assistant Examiner:
Int. Cl.
CPC ...
C07D / ; A61K 3/1517 ;
U.S. Cl.
CPC ...
C07D / ; A61K 3/1517 ;
Abstract
This invention relates generally to the asymmetric synthesis of quinazolin-2-ones that are useful as inhibitors of HIV reverse transcriptase. The synthesis is accomplished through the chiral ligand mediated addition of cyclopropylacetylide.