The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Apr. 01, 2003

Filed:

Oct. 02, 2001
Applicant:
Inventors:

Mukund Shankar Chorghade, Natick, MA (US);

Mukund Keshao Gurjar, Pune, IN;

Palakodety Radha Krishna, Hyderabad, IN;

Sista Venkata Sai Lalitha, Sunnyvale, CA (US);

Kashinath Sadalapure, Dt. Gulbarga, IN;

Susanta Sekhar Adhikari, West Bengal, IN;

Andappan Murugaiah Subbaiah Murugaiah, Tamilnadu, IN;

Sunil Vyankatesh Mhaskar, Natick, MA (US);

Gangavaram Vasantha Madhava Sharma, Hyderabad, IN;

Tangallapally Rajendra Prasad, Warangal, IN;

Punna Sreenivas, Nalgonda, IN;

Vavilala Goverdhan Reddy, Mahabubnagar, IN;

Aminul Islam, Hyderabad, IN;

Chittineni Hari Prasad, Hyderabad, IN;

Alla Venkata Rama Rao, Hyderabad, IN;

Assignee:

Millennium Pharmaceuticals, Inc., Cambridge, MA (US);

Attorney:
Primary Examiner:
Int. Cl.
CPC ...
C07D / ; C07D / ;
U.S. Cl.
CPC ...
C07D / ; C07D / ;
Abstract

The invention includes inter alia new methods for preparation of the pharmaceutically active compound 2-(4-fluorophenoxymethyl)-5-(4-N-hydroxyureidyl-1 -butynyl)-tetrahydrofuran and precursors thereof.


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