The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Sep. 10, 2002

Filed:

Jun. 13, 2000
Applicant:
Inventors:

Christopher F. Bigge, Ann Arbor, MI (US);

Jonathan Wright, Ann Arbor, MI (US);

Sui Xiong Cai, Foothill, CA (US);

Eckard Weber, Laguna Beach, CA (US);

Richard Woodward, Aliso Viejo, CA (US);

Nancy C. Lan, South Pasadena, CA (US);

Zhang-Lin Zhou, Irvine, CA (US);

John F.W. Keana, Eugene, OR (US);

Assignee:

Other;

Attorney:
Primary Examiner:
Int. Cl.
CPC ...
A61K 3/1445 ; C07D / ; C07D / ;
U.S. Cl.
CPC ...
A61K 3/1445 ; C07D / ; C07D / ;
Abstract

Novel 4-substituted piperidine analogs, pharmaceutical compositions containing the same and the method of using the 4-substituted piperidine analogs as selectively active antagonists of N-methyl-D-aspartate (NMDA) receptor subtypes for treating conditions such as cerebral ischemia, central nervous system trauma, hypoglycemia, neurodegenerative disorders, anxiety, migraine headaches, convulsions, aminoglycoside antibiotics-induced hearing loss, chronic pain, psychosis, glaucoma, CMV retinitis, opioid tolerance or withdrawal, urinary incontinence and neurodegenerative disorders such as lathyrism, Alzheimers' Disease, Parkinsonism, and Huntington's Disease are described. Also described are novel methods for preparing 4-substituted piperidine analogs and novel intermediates of the 4-substituted piperidine analogs.


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