The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.
The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.
Patent No.:
Date of Patent:
Aug. 27, 2002
Filed:
Jun. 14, 2001
Hartmut Greiner, Darmstadt, DE;
Gerd Bartoszyk, Weiterstadt, DE;
Henning Böttcher, Darmstadt, DE;
Gerhard Barnickel, Darmstadt, DE;
Bertram Cezanne, Mörfelden-Walldorf, DE;
Merck Patent GmbH, Darmstadt, DE;
Abstract
The present invention relates to sulphonylexazolamines of general formula (I), wherein R , R represent independently from each other H, A, —(CH ) —Ar or alkenyl with 2-6 C atoms, R and R together also represent a mononuclear saturated heterocycle with 1-2 N, O and/or S atoms, Z is H, A, CF , NO , Hal, OH, OA, NH , NHA or NH . A represents alkyl with 1-6 C atoms, Ar is Z-monosubstituted or Z-disubstituted phenyl, Hal is F, Cl, Br, or L n is 1 or 2 of the physiologically acceptable salts or solvates thereof. Said sulphonyloxazolamines are used as therapeutic active ingredients. The invention also relates to the use of sulphonyloxazolamines as therapeutic active ingredients and/or to the production of pharmaceutical preparations to combat diseases of the central nervous system. The invention further relates to a pharmaceutical preparation and the production thereof.