The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Nov. 21, 2000

Filed:

Dec. 11, 1998
Applicant:
Inventors:

Adnan Mjalli, Escondido, CA (US);

Sepehr Sarshar, Cardiff by the Sea, CA (US);

Xiaodong Cao, Carlsbad, CA (US);

Farid Bakir, San Diego, CA (US);

Assignee:

Other;

Attorney:
Primary Examiner:
Assistant Examiner:
Int. Cl.
CPC ...
C07D / ; C07D / ; C07D / ; C07D / ;
U.S. Cl.
CPC ...
548235 ; 548127 ; 548128 ; 548131 ; 548134 ; 548136 ; 548146 ; 548206 ; 548236 ; 548250 ; 548255 ; 5482662 ; 5483351 ; 5483601 ; 5483731 ; 548440 ; 548469 ; 548492 ; 548518 ; 549 60 ; 549 70 ; 549 71 ; 549 72 ; 549414 ; 549425 ; 549426 ; 549429 ; 549430 ; 549434 ; 549462 ; 549483 ; 549484 ; 549491 ; 549398 ; 546152 ; 546167 ; 5462714 ; 544 63 ; 544 83 ; 544 88 ; 544 96 ; 544180 ; 544238 ; 544242 ; 544264 ; 544269 ; 544283 ; 544284 ; 544353 ;
Abstract

The present invention relates to novel protein tyrosine phosphatase modulating compounds having the general structure shown in Formula (A1), to methods for their preparation, to compositions comprising the compounds, to their use for treatment of human and animal disorders, to their use for purification of proteins or glycoproteins, and to their use in diagnosis. The invention relates to modulation of the activity of molecules with phosphotyrosine recognition units, including protein tyrosine phosphatases (PTPases) and proteins with Src-homology-2 domains, in in vitro systems, microorganism, eukaryoic cells, whole animals and human being. R' and R' are independently selected from the group consisting of hydrogen, halo, cyano, nitro, trihalomethyl, alkyl, arylalkyl. R'' is selected from the group consisting of hydrogen, alkyl, substituted alkyl, aryl, arylalkyl. X is aryl. Y is selected from hydrogen or ##STR1## wherein (*) indicates a potential point of attachment to X.


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