The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Mar. 21, 2000

Filed:

May. 28, 1998
Applicant:
Inventors:

Akira Yoshida, Tokyo, JP;

Kozo Oda, Tokyo, JP;

Takashi Kasai, Tokyo, JP;

Kousei Shimada, Tokyo, JP;

Hiroshi Kogen, Tokyo, JP;

Ichiro Hayakawa, Tokyo, JP;

Sadao Ishihara, Tokyo, JP;

Teiichiro Koga, Tokyo, JP;

Eiichi Kitazawa, Tokyo, JP;

Taro Tokui, Tokyo, JP;

Assignee:
Attorney:
Primary Examiner:
Int. Cl.
CPC ...
A61K / ; C07C / ;
U.S. Cl.
CPC ...
514485 ; 560130 ; 560133 ; 560138 ; 564 32 ; 564 47 ; 564 92 ; 564154 ; 564155 ; 564158 ; 514452 ; 514464 ; 514465 ; 514469 ; 514478 ; 514479 ; 514524 ; 514563 ; 514588 ; 514601 ; 514602 ; 514617 ; 514618 ; 514619 ; 549377 ; 549378 ; 549441 ; 549467 ; 549468 ; 554 35 ; 554 36 ; 554 37 ; 554 56 ; 558411 ; 558412 ; 558415 ;
Abstract

Compounds of formula (I): ##STR1## wherein: R.sup.1 is alkyl; R.sup.2a, R.sup.2b, R.sup.2c and R.sup.2d are the same or different and each is hydrogen, optionally substituted alkyl or various other organic groups; R.sup.3 is alkyl; R.sup.4 is a group of formula (II), (III), (IV), (V), (VI), (VII), (VIII) or (IX): ##STR2## wherein: A.sup.1 is a single bond, alkylene or alkenylene; A.sup.2 is or alkenylene; A.sup.3 is a single bond, alkyleneor alkenylene; R.sup.5a and R.sup.5b are the same or different and each is hydrogen, alkyl or various other groups; R.sup.6 is alkyl or phenyl; R.sup.7 is hydrogen or alkyl; R.sup.8 is alkyl or various other groups; and n is 0 and pharmaceutically acceptable salts thereof have valuable inhibitory activity against acyl-CoA: cholesterol acyl transferase.


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