The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Jan. 06, 1998

Filed:

Aug. 05, 1994
Applicant:
Inventors:

Vibhakar J Shah, San Francisco, CA (US);

George L Kenyon, San Francisco, CA (US);

Irwin D Kuntz, Greenbrae, CA (US);

Assignee:
Attorney:
Primary Examiner:
Int. Cl.
CPC ...
C12Q / ; C07H / ; C07K / ; C07K / ;
U.S. Cl.
CPC ...
435-6 ; 435375 ; 435377 ; 536 231 ; 536 243 ; 536 2431 ; 536 2432 ; 536 245 ; 530300 ; 530333 ; 436 86 ; 436 94 ;
Abstract

The present invention provides novel nucleic acid mimics (termed 'PENAMs') comprising a peptidic backbone and nucleotidic sidechains; the sidechains being oriented in such a way that the PENAM is homomorphous to target nucleic acids with which it can effectively hydrogen bond. Homomorphism is achieved by the incorporation of unusual sterochemical centers, including D-chiral centers and quasi-chiral centers, into the peptidic backbone. The PENAMs are useful for targeting nucleic acid sequences in order to modulate their activity in an 'antisense' manner. Targeting can also be used to detect, isolate or modify target nucleic acids.


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