The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Jun. 10, 1997

Filed:

May. 28, 1996
Applicant:
Inventor:

Hubert Maehr, Wayne, NJ (US);

Assignee:

Hoffmann-La Roche Inc., Nutley, NJ (US);

Attorneys:
Primary Examiner:
Int. Cl.
CPC ...
C07F / ;
U.S. Cl.
CPC ...
548119 ; 548205 ;
Abstract

The invention relates to a process of making a compound of the formula ##STR1## wherein R.sub.1, R.sub.2, R.sub.3 and R.sub.4 and n are as described herein, and, when R.sub.1 is different from R.sub.2, and/or when R.sub.3 is different from R.sub.4, enantiomers, diastereomers and racemates thereof, and salts thereof with pharmaceutically acceptable bases. The method comprises reacting a compound of the formula ##STR2## wherein R.sub.5 and n are as described herein with a compound of the formula ##STR3## to produce a compound of the formula ##STR4## wherein n is as described herein, and converting a compound of formula IV to a compound of formula I.


Find Patent Forward Citations

Maehr, Hubert. (1997). Intermediate for (U.S. Patent No. 5637720). U.S. Patent and Trademark Office. https://idiyas.com/patent/badge/5637720

Data source: USPTO (United States Patent and Trademark Office) public patent records. Weekly synchronization. How IDiyas builds this profile

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