The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.
The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.
Patent No.:
Date of Patent:
Nov. 12, 1996
Filed:
Sep. 22, 1994
Applicant:
Inventors:
Michael D Varney, La Costa, CA (US);
Gifford P Marzoni, San Diego, CA (US);
Cynthia L Palmer, La Mesa, CA (US);
Judith P Deal, San Diego, CA (US);
Terence R Jones, San Diego, CA (US);
Assignee:
Agouron Pharmaceuticals, Inc., La Jolla, CA (US);
Primary Examiner:
Int. Cl.
CPC ...
A61K / ; A61K / ; C07D / ; C07D / ;
U.S. Cl.
CPC ...
514257 ; 5142328 ; 514255 ; 514411 ; 544122 ; 544153 ; 544249 ; 544372 ; 548427 ; 548440 ; 548441 ; 548450 ;
Abstract
The invention relates to TS-inhibiting compounds of the formula ##STR1## where W is an alkylene group; D is a structure having two rings that are unsubstituted or substituted, where (i) one ring is a phenyl ring and (ii) the other ring is a phenyl ring or a 6-membered heterocyclic ring; R is a hydrogen atom or an alkyl group; and X and Y together form ##STR2## and to salts of these compounds. The moiety W can be CH.sub.2, and D can be a phenyl ring bridged through a sulfonyl group to another ring.