The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Jul. 02, 1996

Filed:

Jun. 01, 1993
Applicant:
Inventors:

Gunter Neef, Berlin, DE;

Gerald Kirsch, Berlin, DE;

Andreas Stein-Eyer, Berlin, DE;

Katica Schwarz, Berlin, DE;

Matthias Brautigam, Berlin, DE;

Ruth Thieroff-Ekerdt, Berlin, DE;

Petra Rach, Berlin, DE;

Assignee:
Attorney:
Primary Examiner:
Int. Cl.
CPC ...
A61K / ; C07C / ;
U.S. Cl.
CPC ...
514167 ; 552653 ; 540200 ; 540202 ; 544-2 ; 544-3 ; 544 63 ; 544224 ; 546-1 ; 548100 ; 548122 ; 548123 ; 548124 ; 548125 ; 548400 ; 549-1 ; 549 13 ; 549 29 ; 549 88 ;
Abstract

The invention discloses side-chain homologous vitamin D derivatives of formula I ##STR1## in which R.sup.1, R.sup.2, R.sup.3, R.sup.4, R.sup.5, R.sup.6, B, and D have the meanings defined in the specification and either (1) A is a direct bond between carbon atoms 20 and 22 and X is an oxy alkylene radical, --(CH.sub.2).sub.n O-- where n is 1 to 3; (2) A is a methylene bridge, --CH.sub.2 --, between carbon atoms 20 and 22 and X is either an alkylene radical, --(CH.sub.2).sub.n -- or an oxy alkylene radical, --(CH.sub.2).sub.n O--, where n is 1 to 3; or (3) if A is a direct bond and B and D together form a second bond, then X(R.sup.5) (R.sup.6) is ##STR2## The compounds possess proliferation-inhibiting and cell-differentiating activity.


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