The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Mar. 15, 1994

Filed:

Jul. 13, 1989
Applicant:
Inventors:

Heinojo Yamasaka, Ushiku, JP;

Hiroyasu Uchiyama, Koshigaya, JP;

Hirotaka Masuda, Sakura, JP;

Yoshiomi Sakamoto, Oyama, JP;

Yoshimi Nakamigawa, Sekijo, JP;

Mitsuko Yoshioka, Yoshikawa, JP;

Terumasa Moriga, Misato, JP;

Assignee:
Attorney:
Primary Examiner:
Int. Cl.
CPC ...
A61K / ; A61K / ; A61K / ;
U.S. Cl.
CPC ...
424 7801 ; 424451 ; 424452 ; 424456 ; 424463 ; 424464 ; 424465 ; 424474 ; 424480 ; 424485 ; 424486 ; 514212 ; 514338 ; 514395 ; 540603 ; 5483071 ; 546199 ;
Abstract

A stabilized physiologically active benzimidazole derivative having the formula (I): ##STR1## wherein R.sup.1 is hydrogen atom, an alkyl group having 1 to 8 carbon atoms, a fluoroalkyl group having 1 to 6 carbon atoms, a cycloalkyl group, phenyl group or an aralkyl group, R.sup.2 is hydrogen atom or a lower alkyl group, or R.sup.1 and R.sup.2 together with the adjacent nitrogen atom form a ring, and each of R.sup.3a, R.sup.3b, R.sup.4a, R.sup.4b and R.sup.4c independently is hydrogen atom, a halogen atom, a fluoroalkyl group having 1 to 6 carbon atoms, a lower alkyl group, a lower alkoxy group, a lower alkoxycarbonyl group or an amino group. The stabilized benzimidazole derivative is in amorphous form or present in contact with a basic material.


Find Patent Forward Citations

Loading…