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The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Patent No.:

US 5138035 B1

PDFFull Text
Date of Patent:
Aug. 11, 1992

Filed:

Jun. 01, 1990

Cyclopeptide derivatives usable as selective inhibitors with respect to

Applicant:
Inventors:

Michel Wakselman, Paris, FR;

Jean-Paul Mazaleyrate, Choisy-Le-Roi, FR;

Michele Reboud-Ravaux, Paris, FR;

Assignee:

Centre National de la Recherche Scientifique, Paris, FR;

Attorney:

Oblon, Spivak, McClelland, Maier & Neustadt

Primary Examiner:

Merrell C Cashion, Jr

Assistant Examiner:

A M Davenport

Int. Cl.
CPC ...
C07K / ; A61K / ;
U.S. Cl.
CPC ...
530317 ;
Abstract

The invention relates to cyclopeptide derivative usable as protease inhibitors and complying with formula: ##STR1## in which R.sup.1 is a halogen atom, e.g. bromine or a radical such as S.sup.+ R.sub.2.sup.4 X.sub.1/v.sup.v-, R.sup.2 is a hydrogen atom, an alkyl radical, a halogen atom or other groups, R.sup.3 is NH, O or S, Z comprises a peptide sequence Z.sup.1 and a group such that CO has one end connected to the aromatic nucleus and CO-AA is a radical derived fropm an amino acid having a specificity with respect to the protease to be inhibited.

Find Patent Forward Citations

Wakselman, Michel. (1992). Cyclopeptide derivatives usable as selective inhibitors with respect to (U.S. Patent No. 5138035). U.S. Patent and Trademark Office. https://idiyas.com/patent/badge/5138035

Data source: USPTO (United States Patent and Trademark Office) public patent records. Weekly synchronization. How IDiyas builds this profile

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