The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Jul. 10, 1990

Filed:

Nov. 16, 1987
Applicant:
Inventors:

Braham Shroot, Antibes, FR;

Jacques Eustache, Crasse, FR;

Jean-Michel Bernardon, Nice, FR;

Attorney:
Primary Examiner:
Assistant Examiner:
Int. Cl.
CPC ...
A61K / ; A61K / ; A61K / ; A61K / ; C07H / ; C07H / ; C07H / ; C07H / ; C07C / ; C07C / ; C07C / ; C07C / ;
U.S. Cl.
CPC ...
514 62 ; 514319 ; 514423 ; 514730 ; 514859 ; 514863 ; 514885 ; 514886 ; 514880 ; 514887 ; 514912 ; 514 42 ; 514 43 ; 514 63 ; 514532 ; 514533 ; 514543 ; 514546 ; 514547 ; 514548 ; 514549 ; 514550 ; 514551 ; 514569 ; 514617 ; 514618 ; 514621 ; 514622 ; 5142375 ; 514255 ; 546 14 ; 546205 ; 548406 ; 548539 ; 560 56 ; 560 89 ; 560 90 ; 560 91 ; 560100 ; 560194 ; 560250 ; 560251 ; 560252 ; 560255 ; 536 187 ; 536 22 ; 556419 ; 556437 ; 556449 ; 562467 ; 562490 ; 564162 ; 564169 ; 564172 ; 564173 ; 568808 ; 544 64 ; 544176 ; 544225 ; 544391 ;
Abstract

A benzonaphthalene compound has the formula ##STR1## wherein R.sub.1 represents ##STR2## or (ii) --CH.sub.2 OH; R.sub.6 represents ##STR3## or OR.sub.7 wherein R.sub.7 represents hydrogen, alkyl having 1-20 carbon atoms, monohydroxyalkyl or polyhydroxyalkyl, r' or r' represent hydrogen, lower alkyl, mono or polyhydroxyalkyl, aryl or a residue of an amino acid or a sugar, or together form a heterocycle; R.sub.2 represents hydrogen, alkyl having 1-15 carbon atoms, alkoxy having 1-4 carbon atoms or a cycloaliphatic radical; R.sub.3 represents hydrogen, hydroxy, alkyl having 1-4 carbon atoms, alkoxy having 1-10 carbon atoms, a cycloaliphatic radical, a thiocycloaliphatic radical or --O--Si(CH.sub.3).sub.2 --R.sub.8 wherein R.sub.8 represents lower alkyl; and R.sub.4 and R.sub.5 represent hydrogen, lower alkyl, hydroxy or lower acyloxy. This compound is useful in the topical and systemic treatment of dermatologic diseases and in the treatment of the degeneration of conjunctive tissues. The compound also possesses anti-tumor acitivity.


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