The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Jul. 28, 1987

Filed:

Jan. 22, 1985
Applicant:
Inventors:

Karin M Kirkland, Wilmington, DE (US);

Derrick M Mant, Stockport, GB;

Assignees:

ICI Americas Inc., Wilmington, DE (US);

Imperial Chemical Industries PLC, London, GB;

Attorney:
Primary Examiner:
Assistant Examiner:
Int. Cl.
CPC ...
A61K / ; A61K / ; C07D / ; C07D / ;
U.S. Cl.
CPC ...
514211 ; 514212 ; 514218 ; 514228 ; 514230 ; 514233 ; 514241 ; 514242 ; 514245 ; 514252 ; 514269 ; 514272 ; 514274 ; 514316 ; 514318 ; 514326 ; 514340 ; 514341 ; 514359 ; 514361 ; 514362 ; 514363 ; 514364 ; 514365 ; 514369 ; 514370 ; 514372 ; 514374 ; 514376 ; 514377 ; 514378 ; 514380 ; 514383 ; 514384 ; 514385 ; 514397 ; 514398 ; 514402 ; 514403 ; 514406 ; 514407 ; 540544 ; 540553 ; 540575 ; 540596 ; 540597 ; 540598 ; 540601 ; 540602 ; 540603 ; 544-2 ; 544-3 ; 544-7 ; 544-8 ; 544 55 ; 544 56 ; 544 586 ; 544 63 ; 544 66 ; 544 67 ; 544 72 ; 544 82 ; 544 96 ; 544 98 ; 544111 ; 544112 ; 544113 ; 544114 ; 544120 ; 544121 ; 544122 ; 544124 ; 544130 ; 544131 ; 544132 ; 544133 ; 544134 ; 544137 ; 544138 ; 544139 ; 544140 ; 544141 ; 544180 ; 544182 ; 544194 ; 544212 ; 544213 ; 544216 ; 544217 ; 544218 ; 544219 ; 544224 ; 544238 ; 544242 ; 544295 ; 544296 ; 544298 ; 544315 ; 544316 ; 544317 ; 544319 ; 544320 ; 544322 ; 544324 ; 544326 ; 544327 ; 544328 ; 544329 ; 544330 ; 544331 ; 544332 ; 544333 ; 544336 ; 544357 ; 544358 ; 544544360 ; 544364 ; 544366 ; 544367 ; 544369 ; 544370 ; 544371 ; 544372 ; 544405 ; 546187 ; 546193 ; 546208 ; 546209 ; 546210 ; 546211 ; 546255 ; 546256 ; 546264 ; 546275 ; 546276 ; 546277 ; 546278 ; 546279 ; 546280 ; 546281 ; 546283 ; 546284 ; 546306 ; 546332 ; 548125 ; 548127 ; 548128 ; 548129 ; 548130 ; 548548132 ; 548133 ; 548134 ; 548135 ; 548136 ; 548138 ; 548141 ; 548143 ; 548144 ; 548146 ; 548182 ; 548183 ; 548184 ; 548187 ; 548190 ; 548191 ; 548194 ; 548206 ; 548213 ; 548214 ; 548215 ; 548225 ; 548226 ; 548227 ; 548228 ; 548229 ; 548230 ; 548232 ; 548233 ; 548240 ; 548243 ; 548244 ; 548245 ; 548246 ; 548247 ; 548249 ; 548255 ; 548262 ; 548264 ; 548265 ; 548266 ; 548267 ; 548269 ; 548300 ; 548336 ; 548337 ; 548342 ; 548348 ; 548356 ; 548375 ; 548376 ; 548377 ; 548378 ; 548379 ; 548517 ; 548518 ; 548519 ; 548521 ; 548527 ; 548540 ; 548541 ; 548543 ; 548544 ; 548550 ; 548557 ; 548558 ;
Abstract

A guanidine derivative of the formula I: ##STR1## in which R.sup.1, R.sup.2, R.sup.3, R.sup.4, ring X and D are a variety of radicals defined in the specification and A is a 3-8C alkylene chain which is substituted by a hydroxy radical and into which is optionally inserted, as part of the backbone of the chain, one or two groups selected from oxygen and sulphur atoms and NH and 1-6C N-alkyl radicals; and the pharmaceutically-acceptable acid additions salts thereof. Pharmaceutical compositions and methods of manufacture are also described. The compound of the formula I is a histamine H-2 antagonist and is therefore useful in ulcer therapy.


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