The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Feb. 18, 1986

Filed:

May. 16, 1984
Applicant:
Inventors:

John M Evans, Roydon, GB;

Frederick Cassidy, Harlow, GB;

Assignee:
Attorney:
Primary Examiner:
Int. Cl.
CPC ...
A61K / ; C07D / ;
U.S. Cl.
CPC ...
514456 ; 514242 ; 514241 ; 514444 ; 549404 ; 549399 ; 514443 ; 549345 ; 549 60 ; 514422 ; 549 57 ; 549 55 ; 514414 ; 549 54 ; 549 52 ; 514409 ; 549 51 ; 548525 ; 514397 ; 548454 ; 548407 ; 514380 ; 548336 ; 548236 ; 514378 ; 548216 ; 548214 ; 514377 ; 548213 ; 548189 ; 514376 ; 548188 ; 548147 ; 514374 ; 548136 ; 548134 ; 514372 ; 548130 ; 548129 ; 514371 ; 548128 ; 548127 ; 514370 ; 546269 ; 544405 ; 514369 ; 544333 ; 544298 ; 514365 ; 544240 ; 544239 ; 514363 ; 544238 ; 544230 ; 514362 ; 514361 ; 514337 ; 514314 ; 514313 ; 514312 ; 514307 ; 514278 ; 514275 ; 514274 ; 514272 ; 514269 ; 514256 ; 514255 ; 514247 ;
Abstract

Compounds of formula (I): ##STR1## wherein: either one of R.sub.1 and R.sub.2 is hydrogen and the other is selected from the class of C.sub.1-6 alkylcarbonyl, C.sub.1-6 alkoxycarbonyl, C.sub.1-6 alkylcarbonyloxy, C.sub.1-6 alkylhydroxymethyl, nitro, cyano, chloro, trifluoromethyl, C.sub.1-6 alkylsulphinyl, C.sub.1-6 alkylsulphonyl, C.sub.1-6 alkoxysulphinyl, C.sub.1-6 alkoxysulphonyl, C.sub.1-6 alkylcarbonylamino, C.sub.1-6 alkoxycarbonylamino, C.sub.1-6 alkyl-thiocarbonyl, C.sub.1-6 alkoxy-thiocarbonyl, C.sub.1-6 alkyl-thiocarbonyloxy, 1-mercapto C.sub.2-7 alkyl, formyl or aminosulphinyl, aminosulphonyl or aminocarbonyl, the amino moiety being optionally substituted by one or two C.sub.1-6 alkyl groups, or C.sub.1-6 alkylsulphinylamino, C.sub.1-6 alkylsulphonylamino C.sub.1-6 alkoxysulphinylamino or C.sub.1-6 alkoxysulphonylamino, or ethylenyl terminally substituted by C.sub.1-6 alkylcarbonyl, nitro or cyano, or --C(C.sub.1-6 alkyl)NOH or --C(C.sub.1-6 alkyl)NNH.sub.2, or one of R.sub.1 and R.sub.2 is nitro, cyano or C.sub.1-3 alkylcarbonyl and the other is methoxy or amino optionally substituted by one or two C.sub.1-6 alkyl or by C.sub.2-7 alkanoyl;


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