The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.

The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.

Date of Patent:
Feb. 21, 1984

Filed:

Oct. 22, 1981
Applicant:
Inventor:

Francois Picart, Dijon, FR;

Attorney:
Primary Examiner:
Int. Cl.
CPC ...
A61K / ; C07H / ;
U.S. Cl.
CPC ...
424180 ; 536-41 ; 536 179 ; 536 176 ; 536 178 ;
Abstract

The present invention relates to the benzoyl- and .alpha.-hydroxybenzyl-phenyl-oside derivatives of general formula: ##STR1## [in which Z is CO or CHOH, X.sub.1, X.sub.2, X.sub.3, X.sub.4 and X.sub.5, which are identical or different, each represent an atom of hydrogen, an atom of halogen, an alkyl group with 1 to 4 carbon atoms, an alkyl group with 1 to 4 carbon atoms substituted by one or more atoms of halogen, an OH group, an alkoxy group with 1 to 4 carbon atoms, an alkoxy group with 1 to 4 carbon atoms, substituted by one or more atoms of halogen, a nitro group, a cyano group, a thiocyano group, an isothiocyano group, a NR'R' group (where R' and R', identical or different, each represent an atom of hydrogen or an alkyl group with 1 to 4 carbon atoms) X.sub.1 being able, in addition, to represent an --NH--CS--O--CH.sub.3 group or an --O--C(CH.sub.3).sub.2 CO.sub.2 --R'' group (where R'' is an alkyl group with 1 to 4 carbon atoms and, preferably, an isopropyl group); and R represents a radical ose (the hydroxyl and amine functions of the radical ose being able to be substituted by acyl, alkyl or sulfate groups)], and to their diastereoisomers. It also relates to the method for preparing these derivatives and to their application in therapeutics.


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