The patent badge is an abbreviated version of the USPTO patent document. The patent badge does contain a link to the full patent document.
The patent badge is an abbreviated version of the USPTO patent document. The patent badge covers the following: Patent number, Date patent was issued, Date patent was filed, Title of the patent, Applicant, Inventor, Assignee, Attorney firm, Primary examiner, Assistant examiner, CPCs, and Abstract. The patent badge does contain a link to the full patent document (in Adobe Acrobat format, aka pdf). To download or print any patent click here.
Patent No.:
Date of Patent:
Dec. 01, 1981
Filed:
Mar. 08, 1978
Syoji Ono, Kodaira, JP;
Takashi Sugiyama, Tokyo, JP;
Yoshiko Kawakami, Higashiyamato, JP;
Yataro Ichikawa, Fuchu, JP;
Yoji Suzuki, Hino, JP;
Hitoshi Ohmori, Hino, JP;
Akiko Azuma, Kodaira, JP;
Teijin Limited, Osaka, JP;
Abstract
This invention provides novel penicillin derivatives of formula [I]; ##STR1## wherein A is hydrogen or hydroxyl, and B represents the cumarin nucleus of formula [III-a]; ##STR2## in which B.sub.1, B.sub.2, B.sub.3, B.sub.4 and B.sub.5 are same or different, and are hydrogen or substituent groups that may contain nitrogen, sulfur or oxygen atom, or nontoxic salts thereof, and bactericides containing said novel penicillin derivatives or nontoxic salts thereof as the main ingredient, and also an advantageous process for producing said novel penicillin derivatives or nontoxic salts thereof, which comprises reacting a derivative of .alpha.-aminobenzylpenicillin with a coumarincarboxylic acid or reacting 6-aminopencillanic acid, a carboxylic acid salt thereof or a protected derivative thereof having the carboxyl blocked with a readily removable protecting group, with a coumarincarboxylic acid phenylglycinamide.